By Kenneth H. Lundstrom (Editor), Mark L. Chiu (Editor)
The extensive diversity of G protein-coupled receptors (GPCRs) encompasses all components of contemporary drugs and feature a massive effect at the strategy of drug improvement. utilizing disease-oriented how to conceal every little thing from screening to expression and crystallization, G Protein-Coupled Receptors in Drug Discovery describes the physiological roles of GPCRs and their involvement in quite a few human ailments. The e-book offers present techniques in drug discovery that come with goal choice, institution of screening and sensible assays. It additionally covers recombinant GPCR expression for drug screening and structural biology, diversified tools for structural characterization of GPCRs, and the significance of bioinformatics. The e-book has been rigorously edited to prevent overlapping info, a few duplication has been deliberately accepted in order that every one bankruptcy can functionality as an self sustaining unit. delivering in-depth discussions on constitution and dynamics of GPCRs, this publication outlines the significance of the GPCRs to drug discovery regularly and drug goals particularly. Daniel E. Levy, editor of the Drug Discovery sequence, is the founding father of DEL BioPharma, a consulting carrier for drug discovery courses. He additionally keeps a weblog that explores natural chemistry.
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Additional resources for G Protein-Coupled Receptors in Drug Discovery
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